Cytoplasmic Dynein Antagonists with Improved Potency and Isoform Selectivity

November 11th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00895

[Cu(o-phthalate)(phenanthroline)] Exhibits Unique Superoxide-Mediated NCI-60 Chemotherapeutic Action through Genomic DNA Damage and Mitochondrial Dysfunction

November 10th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00513
  • Posted in ACS Chemical Biology, Publications
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Switching the Regioselectivity of a Cyclohexanone Monooxygenase toward (+)-trans-Dihydrocarvone by Rational Protein Design

November 9th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00723
  • Posted in ACS Chemical Biology, Publications
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PDZ-Reactive Peptide Activates Ephrin-B Reverse Signaling and Inhibits Neuronal Chemotaxis

November 9th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00889

Small Molecule Microarrays Enable the Identification of a Selective, Quadruplex-Binding Inhibitor of MYC Expression

November 6th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00577
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Conversion of a Single Polypharmacological Agent into Selective Bivalent Inhibitors of Intracellular Kinase Activity

November 6th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00847
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Self-Assembling NanoLuc Luciferase Fragments as Probes for Protein Aggregation in Living Cells

November 6th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00758

Wall teichoic acids prevent antibody binding to epitopes within the cell wall of Staphylococcus aureus

November 5th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00439
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Single-Cell, Time-Resolved Antimicrobial Effects of a Highly Cationic, Random Nylon-3 Copolymer on Live Escherichia coli

November 5th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00547
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Chemical Tools for the Study of Intramembrane Proteases

November 5th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00693