Small Molecules for Cell Reprogramming and Heart Repair: Progress and Perspective

January 6th, 2014 by Min Xie, Nan Cao and Sheng Ding

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ACS Chemical Biology
DOI: 10.1021/cb400865w

Quinine Dimers Are Potent Inhibitors of the Plasmodium falciparum Chloroquine Resistance Transporter and Are Active against Quinoline-Resistant P. falciparum

January 5th, 2014 by Christine A. Hrycyna, Robert L. Summers, Adele M. Lehane, Marcos M. Pires, Hilda Namanja, Kelsey Bohn, Jerrin Kuriakose, Michael Ferdig, Philipp P. Henrich, David A. Fidock, Kiaran Kirk, Jean Chmielewski and Rowena E. Martin

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ACS Chemical Biology
DOI: 10.1021/cb4008953
  • Posted in ACS Chemical Biology, Publications
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Targeting the Production of Oncogenic MicroRNAs with Multimodal Synthetic Small Molecules

January 3rd, 2014 by Duc Duy Vo, Cathy Staedel, Laura Zehnacker, Rachid Benhida, Fabien Darfeuille and Maria Duca

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ACS Chemical Biology
DOI: 10.1021/cb400668h

Context Clues: The Importance of Stem Cell–Material Interactions

January 3rd, 2014 by Andrew S. Khalil, Angela W. Xie and William L. Murphy

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ACS Chemical Biology
DOI: 10.1021/cb400801m

Ligand-Independent and Tissue-Selective Androgen Receptor Inhibition by Pyrvinium

January 3rd, 2014 by Minyoung Lim, Maya Otto-Duessel, Miaoling He, Leila Su, Dan Nguyen, Emily Chin, Tamara Alliston and Jeremy O. Jones

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ACS Chemical Biology
DOI: 10.1021/cb400759d

Distinct BimBH3 (BimSAHB) Stapled Peptides for Structural and Cellular Studies

January 2nd, 2014 by Greg H. Bird, Evripidis Gavathiotis, James L. LaBelle, Samuel G. Katz and Loren D. Walensky

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ACS Chemical Biology
DOI: 10.1021/cb4003305

Identification and Validation of Cryptochrome Inhibitors That Modulate the Molecular Circadian Clock

January 2nd, 2014 by Sung Kook Chun, Jaebong Jang, Sooyoung Chung, Hwayoung Yun, Nam-Jung Kim, Jong-Wha Jung, Gi Hoon Son, Young-Ger Suh and Kyungjin Kim

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ACS Chemical Biology
DOI: 10.1021/cb400752k
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Chemical Synthesis of Insulin Analogs through a Novel Precursor

January 2nd, 2014 by Alexander N. Zaykov, John P. Mayer, Vasily M. Gelfanov and Richard D. DiMarchi

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ACS Chemical Biology
DOI: 10.1021/cb400792s

Long Residence Time Inhibition of EZH2 in Activated Polycomb Repressive Complex 2

December 31st, 2013 by Glenn S. Van Aller, Melissa Baker Pappalardi, Heidi M. Ott, Elsie Diaz, Martin Brandt, Benjamin J. Schwartz, William H. Miller, Dashyant Dhanak, Michael T. McCabe, Sharad K. Verma, Caretha L. Creasy, Peter J. Tummino and Ryan G. Kruger

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ACS Chemical Biology
DOI: 10.1021/cb4008748

Pre-mRNA Splicing-Modulatory Pharmacophores: The Total Synthesis of Herboxidiene, a Pladienolide–Herboxidiene Hybrid Analog and Related Derivatives

December 30th, 2013 by Chandraiah Lagisetti, Maria V. Yermolina, Lalit Kumar Sharma, Gustavo Palacios, Brett J. Prigaro and Thomas R. Webb

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ACS Chemical Biology
DOI: 10.1021/cb400695j
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