Ligand-Independent and Tissue-Selective Androgen Receptor Inhibition by Pyrvinium

January 3rd, 2014 by Minyoung Lim, Maya Otto-Duessel, Miaoling He, Leila Su, Dan Nguyen, Emily Chin, Tamara Alliston and Jeremy O. Jones

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ACS Chemical Biology
DOI: 10.1021/cb400759d

Distinct BimBH3 (BimSAHB) Stapled Peptides for Structural and Cellular Studies

January 2nd, 2014 by Greg H. Bird, Evripidis Gavathiotis, James L. LaBelle, Samuel G. Katz and Loren D. Walensky

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ACS Chemical Biology
DOI: 10.1021/cb4003305

Identification and Validation of Cryptochrome Inhibitors That Modulate the Molecular Circadian Clock

January 2nd, 2014 by Sung Kook Chun, Jaebong Jang, Sooyoung Chung, Hwayoung Yun, Nam-Jung Kim, Jong-Wha Jung, Gi Hoon Son, Young-Ger Suh and Kyungjin Kim

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ACS Chemical Biology
DOI: 10.1021/cb400752k
  • Posted in ACS Chemical Biology, Publications
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Chemical Synthesis of Insulin Analogs through a Novel Precursor

January 2nd, 2014 by Alexander N. Zaykov, John P. Mayer, Vasily M. Gelfanov and Richard D. DiMarchi

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ACS Chemical Biology
DOI: 10.1021/cb400792s

Long Residence Time Inhibition of EZH2 in Activated Polycomb Repressive Complex 2

December 31st, 2013 by Glenn S. Van Aller, Melissa Baker Pappalardi, Heidi M. Ott, Elsie Diaz, Martin Brandt, Benjamin J. Schwartz, William H. Miller, Dashyant Dhanak, Michael T. McCabe, Sharad K. Verma, Caretha L. Creasy, Peter J. Tummino and Ryan G. Kruger

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ACS Chemical Biology
DOI: 10.1021/cb4008748

Pre-mRNA Splicing-Modulatory Pharmacophores: The Total Synthesis of Herboxidiene, a Pladienolide–Herboxidiene Hybrid Analog and Related Derivatives

December 30th, 2013 by Chandraiah Lagisetti, Maria V. Yermolina, Lalit Kumar Sharma, Gustavo Palacios, Brett J. Prigaro and Thomas R. Webb

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ACS Chemical Biology
DOI: 10.1021/cb400695j
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Defining Binding Efficiency and Specificity of Auxins for SCFTIR1/AFB-Aux/IAA Co-receptor Complex Formation

December 23rd, 2013 by Sarah Lee, Shanthy Sundaram, Lynne Armitage, John P. Evans, Tim Hawkes, Stefan Kepinski, Noel Ferro and Richard M. Napier

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ACS Chemical Biology
DOI: 10.1021/cb400618m
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Auranofin Is an Apoptosis-Simulating Agent with in Vitro and in Vivo Anti-leishmanial Activity

December 23rd, 2013 by Elizabeth R. Sharlow, Stephanie Leimgruber, Samantha Murray, Ana Lira, Richard J. Sciotti, Mark Hickman, Thomas Hudson, Susan Leed, Diana Caridha, Amy M. Barrios, David Close, Max Grögl and John S. Lazo

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ACS Chemical Biology
DOI: 10.1021/cb400800q

Dual Labeling of Lipopolysaccharides for SPECT-CT Imaging and Fluorescence Microscopy

December 20th, 2013 by Vincent Duheron, Mathieu Moreau, Bertrand Collin, Wahib Sali, Claire Bernhard, Christine Goze, Thomas Gautier, Jean-Paul Pais de Barros, Valérie Deckert, François Brunotte, Laurent Lagrost and Franck Denat

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ACS Chemical Biology
DOI: 10.1021/cb400779j

Time- and Concentration-Dependent Effects of Exogenous Serotonin and Inflammatory Cytokines on Mast Cell Function

December 19th, 2013 by Sarah M. Gruba, Audrey F. Meyer, Benjamin M. Manning, Yiwen Wang, John W. Thompson, Joseph J. Dalluge and Christy L. Haynes

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ACS Chemical Biology
DOI: 10.1021/cb400787s
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