Acetyl-lysine Binding Site of Bromodomain-Containing Protein 4 (BRD4) Interacts with Diverse Kinase Inhibitors

March 13th, 2014 by Stuart W. J. Ember, Jin-Yi Zhu, Sanne H. Olesen, Mathew P. Martin, Andreas Becker, Norbert Berndt, Gunda I. Georg and Ernst Schönbrunn

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ACS Chemical Biology
DOI: 10.1021/cb500072z
  • Posted in ACS Chemical Biology, Publications
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Molecular Determinants of a Regulatory Prolyl Isomerization in the Signal Adapter Protein c-CrkII

March 10th, 2014 by Philipp A. M. Schmidpeter and Franz X. Schmid

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ACS Chemical Biology
DOI: 10.1021/cb500001n
  • Posted in ACS Chemical Biology, Publications
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A Structural and Energetic Model for the Slow-Onset Inhibition of the Mycobacterium tuberculosis Enoyl-ACP Reductase InhA

March 10th, 2014 by Huei-Jiun Li, Cheng-Tsung Lai, Pan Pan, Weixuan Yu, Nina Liu, Gopal R. Bommineni, Miguel Garcia-Diaz, Carlos Simmerling and Peter J. Tonge

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ACS Chemical Biology
DOI: 10.1021/cb400896g
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Organophosphorus Flame Retardants Inhibit Specific Liver Carboxylesterases and Cause Serum Hypertriglyceridemia

March 10th, 2014 by Patrick J. Morris, Daniel Medina-Cleghorn, Ann Heslin, Sarah M. King, Joseph Orr, Melinda M. Mulvihill, Ronald M. Krauss and Daniel K. Nomura

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ACS Chemical Biology
DOI: 10.1021/cb500014r
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Cyclic Nucleotide Mapping of Hyperpolarization-Activated Cyclic Nucleotide-Gated (HCN) Channels

March 7th, 2014 by Stefan Möller, Andrea Alfieri, Daniela Bertinetti, Marco Aquila, Frank Schwede, Marco Lolicato, Holger Rehmann, Anna Moroni and Friedrich W. Herberg

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ACS Chemical Biology
DOI: 10.1021/cb400904s

MVAPACK: A Complete Data Handling Package for NMR Metabolomics

March 7th, 2014 by Bradley Worley and Robert Powers

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ACS Chemical Biology
DOI: 10.1021/cb4008937

Insights into the Biosynthesis of 12-Membered Resorcylic Acid Lactones from Heterologous Production in Saccharomyces cerevisiae

March 6th, 2014 by Yuquan Xu, Tong Zhou, Patricia Espinosa-Artiles, Ying Tang, Jixun Zhan and István Molnár

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ACS Chemical Biology
DOI: 10.1021/cb500043g
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Selective Ligand Behaviors Provide New Insights into Agonist Activation of Nicotinic Acetylcholine Receptors

March 5th, 2014 by Christopher B. Marotta, Iva Rreza, Henry A. Lester and Dennis A. Dougherty

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ACS Chemical Biology
DOI: 10.1021/cb400937d
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A Key n→π* Interaction in N-Acyl Homoserine Lactones

February 26th, 2014 by Robert W. Newberry and Ronald T. Raines

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ACS Chemical Biology
DOI: 10.1021/cb500022u

Imparting Albumin-Binding Affinity to a Human Protein by Mimicking the Contact Surface of a Bacterial Binding Protein

February 26th, 2014 by Satoshi Oshiro and Shinya Honda

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ACS Chemical Biology
DOI: 10.1021/cb400946m
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