Boronic Acid for the Traceless Delivery of Proteins into Cells

December 15th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00966

Mitochondria-Targeted Approach: Remarkably Enhanced Cellular Bioactivities of TPP2a as Selective Inhibitor and Probe toward TrxR

December 14th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00708
  • Posted in ACS Chemical Biology, Publications
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Three Residues Make an Evolutionary Switch for Folding and RNA-Destabilizing Activity in the TTP Family of Proteins

December 14th, 2015 by Laura M. Deveau and Francesca Massi

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00639
  • Posted in ACS Chemical Biology, Publications
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Azacyclic FTY720 Analogues That Limit Nutrient Transporter Expression but Lack S1P Receptor Activity and Negative Chronotropic Effects Offer a Novel and Effective Strategy to Kill Cancer Cells in Vivo

December 14th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00761
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Thiostrepton Variants Containing a Contracted Quinaldic Acid Macrocycle Result from Mutagenesis of the Second Residue

December 14th, 2015 by Feifei Zhang, Chaoxuan Li and Wendy L. Kelly

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00731
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NanoLuc Complementation Reporter Optimized for Accurate Measurement of Protein Interactions in Cells

December 10th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00753
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Barrel-shaped ClpP Proteases Display Attenuated Cleavage Specificities

December 9th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00757

A Potent, Selective, and Cell-Active Inhibitor of Human Type I Protein Arginine Methyltransferases

December 8th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00839
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In Vivo Detection of Mitochondrial Dysfunction Induced by Clinical Drugs and Disease-Associated Genes Using a Novel Dye ZMJ214 in Zebrafish

December 8th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00751
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Small Molecule Targeting of a MicroRNA Associated with Hepatocellular Carcinoma

December 7th, 2015 by Jessica L. Childs-Disney and Matthew D. Disney

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00615