Phosphatase-Inert Glucosamine 6-Phosphate Mimics Serve as Actuators of the glmS Riboswitch

October 27th, 2014 by Xiang Fei, Thomas Holmes, Julianna Diddle, Lauren Hintz, Dan Delaney, Alex Stock, Danielle Renner, Molly McDevitt, David B. Berkowitz and Juliane K. Soukup

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ACS Chemical Biology
DOI: 10.1021/cb500458f

DFG-out Mode of Inhibition by an Irreversible Type-1 Inhibitor Capable of Overcoming Gate-Keeper Mutations in FGF Receptors

October 27th, 2014 by Zhifeng Huang, Li Tan, Huiyan Wang, Yang Liu, Steven Blais, Jingjing Deng, Thomas A. Neubert, Nathanael S. Gray, Xiaokun Li and Moosa Mohammadi

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ACS Chemical Biology
DOI: 10.1021/cb500674s
  • Posted in ACS Chemical Biology, Publications
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Fluorinated Aromatic Amino Acids Are Sensitive 19F NMR Probes for Bromodomain-Ligand Interactions

October 27th, 2014 by Neeraj K. Mishra, Andrew K. Urick, Stuart W. J. Ember, Ernst Schönbrunn and William C. Pomerantz

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ACS Chemical Biology
DOI: 10.1021/cb5007344
  • Posted in ACS Chemical Biology, Publications
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Competitive Binding of a Benzimidazole to the Histone-Binding Pocket of the Pygo PHD Finger

October 24th, 2014 by Thomas C. R. Miller, Trevor J. Rutherford, Kristian Birchall, Jasveen Chugh, Marc Fiedler and Mariann Bienz

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ACS Chemical Biology
DOI: 10.1021/cb500585s

Reconstruction of Cladoniamide Biosynthesis Reveals Nonenzymatic Routes to Bisindole Diversity

October 24th, 2014 by Yi-Ling Du, David E. Williams, Brian O. Patrick, Raymond J. Andersen and Katherine S. Ryan

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ACS Chemical Biology
DOI: 10.1021/cb500728h

Dynamic Principle for Designing Antagonistic/Agonistic Molecules for EphA4 Receptor, the Only Known ALS Modifier

October 23rd, 2014 by Haina Qin, Liang-Zhong Lim and Jianxing Song

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ACS Chemical Biology
DOI: 10.1021/cb500413n
  • Posted in ACS Chemical Biology, Publications
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Correction to Recent Mechanistic Insights on Glycoconjugate Vaccines and Future Perspectives

October 23rd, 2014 by Francesco Berti and Roberto Adamo

ACS Chemical Biology
DOI: 10.1021/cb500822h

Recent Progress in Design of Protein-Based Fluorescent Biosensors and Their Cellular Applications

October 23rd, 2014 by Tomonori Tamura and Itaru Hamachi

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ACS Chemical Biology
DOI: 10.1021/cb500661v
  • Posted in ACS Chemical Biology, Publications
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Clickable Analogue of Cerulenin as Chemical Probe to Explore Protein Palmitoylation

October 23rd, 2014 by Baohui Zheng, Shunying Zhu and Xu Wu

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ACS Chemical Biology
DOI: 10.1021/cb500758s

Lipid-Dependent Bimodal MCL1 Membrane Activity

October 22nd, 2014 by Olatz Landeta, Juan GarciaValero, Hector Flores-Romero, Itsasne Bustillo-Zabalbeitia, Ane Landajuela, Miguel Garcia-Porras, Oihana Terrones and Gorka Basañez

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ACS Chemical Biology
DOI: 10.1021/cb500592e