Subtype-Specific Modulation of Estrogen Receptor–Coactivator Interaction by Phosphorylation

November 11th, 2014 by Inga M. Tharun, Lidia Nieto, Christian Haase, Marcel Scheepstra, Mark Balk, Sabine Möcklinghoff, Wencke Adriaens, Sonja A. Dames and Luc Brunsveld

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ACS Chemical Biology
DOI: 10.1021/cb5007097

Time-Resolved FRET Binding Assay to Investigate Hetero-Oligomer Binding Properties: Proof of Concept with Dopamine D1/D3 Heterodimer

November 11th, 2014 by Candide Hounsou, Jean-François Margathe, Nadia Oueslati, Abderazak Belhocine, Elodie Dupuis, Cécile Thomas, André Mann, Brigitte Ilien, Didier Rognan, Eric Trinquet, Marcel Hibert, Jean-Philippe Pin, Dominique Bonnet and Thierry Durroux

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ACS Chemical Biology
DOI: 10.1021/cb5007568
  • Posted in ACS Chemical Biology, Publications
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Regulation of Wnt Signaling Target Gene Expression by the Histone Methyltransferase DOT1L

November 10th, 2014 by Garrett S. Gibbons, Scott R. Owens, Eric R. Fearon and Zaneta Nikolovska-Coleska

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ACS Chemical Biology
DOI: 10.1021/cb500668u

Peptide-Based, Two-Fluorophore, Ratiometric Probe for Quantifying Mobile Zinc in Biological Solutions

November 10th, 2014 by Daniel Y. Zhang, Maria Azrad, Wendy Demark-Wahnefried, Christopher J. Frederickson, Stephen J. Lippard and Robert J. Radford

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ACS Chemical Biology
DOI: 10.1021/cb500617c
  • Posted in ACS Chemical Biology, Publications
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One-Step Enzymatic Modification of the Cell Surface Redirects Cellular Cytotoxicity and Parasite Tropism

November 10th, 2014 by Lee Kim Swee, Sebastian Lourido, George W. Bell, Jessica R. Ingram and Hidde L. Ploegh

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ACS Chemical Biology
DOI: 10.1021/cb500462t
  • Posted in ACS Chemical Biology, Publications
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Multicolor Monitoring of the Proteasome’s Catalytic Signature

November 7th, 2014 by Melanie A. Priestman, Qunzhao Wang, Finith E. Jernigan, Ruma Chowdhury, Marion Schmidt and David S. Lawrence

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ACS Chemical Biology
DOI: 10.1021/cb5007322

Changing the Selectivity of p300 by Acetyl-CoA Modulation of Histone Acetylation

November 6th, 2014 by Ryan A. Henry, Yin-Ming Kuo, Vikram Bhattacharjee, Timothy J. Yen and Andrew J. Andrews

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ACS Chemical Biology
DOI: 10.1021/cb500726b

Distant Polypharmacology among MLP Chemical Probes

November 6th, 2014 by Albert A. Antolín and Jordi Mestres

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ACS Chemical Biology
DOI: 10.1021/cb500393m

Unified and Isomer-Specific NMR Metabolomics Database for the Accurate Analysis of 13C–1H HSQC Spectra

November 5th, 2014 by Kerem Bingol, Da-Wei Li, Lei Bruschweiler-Li, Oscar A. Cabrera, Timothy Megraw, Fengli Zhang and Rafael Brüschweiler

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ACS Chemical Biology
DOI: 10.1021/cb5006382
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Chemical Genetics Screening Reveals KIAA1363 as a Cytokine-Lowering Target

November 5th, 2014 by Devon M. Hunerdosse, Patrick J. Morris, David K. Miyamoto, Karl J. Fisher, Leslie A. Bateman, Jonathan R. Ghazaleh, Sharon Zhong and Daniel K. Nomura

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ACS Chemical Biology
DOI: 10.1021/cb500717g