The Elastase-PK101 Structure: Mechanism of an Ultrasensitive Activity-based Probe Revealed

January 22nd, 2015 by Bernhard C. Lechtenberg, Paulina Kasperkiewicz, Howard Robinson, Marcin Drag and Stefan J. Riedl

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ACS Chemical Biology
DOI: 10.1021/cb500909n

Critical Evaluation and Rate Constants of Chemoselective Ligation Reactions for Stoichiometric Conjugations in Water

January 22nd, 2015 by Fumito Saito, Hidetoshi Noda and Jeffrey W. Bode

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ACS Chemical Biology
DOI: 10.1021/cb5006728
  • Posted in ACS Chemical Biology, Publications
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Structural and Functional Analysis of the Loading Acyltransferase from Avermectin Modular Polyketide Synthase

January 22nd, 2015 by Fen Wang, Yanjie Wang, Junjie Ji, Zhan Zhou, Jingkai Yu, Hua Zhu, Zhiguo Su, Lixin Zhang and Jianting Zheng

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ACS Chemical Biology
DOI: 10.1021/cb500873k
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Chemical Cross-Linking/Mass Spectrometry Maps the Amyloid β Peptide Binding Region on Both Apolipoprotein E Domains

January 21st, 2015 by Stéphanie Deroo, Florian Stengel, Azadeh Mohammadi, Nicolas Henry, Ellen Hubin, Eva-Maria Krammer, Ruedi Aebersold and Vincent Raussens

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ACS Chemical Biology
DOI: 10.1021/cb500994j
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Modulation of Alternative Splicing with Chemical Compounds in New Therapeutics for Human Diseases

January 20th, 2015 by Kenji Ohe and Masatoshi Hagiwara

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ACS Chemical Biology
DOI: 10.1021/cb500697f
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Saturation Mutagenesis of TsrA Ala4 Unveils a Highly Mutable Residue of Thiostrepton A

January 20th, 2015 by Feifei Zhang and Wendy L. Kelly

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ACS Chemical Biology
DOI: 10.1021/cb5007745

Ironing out Their Differences: Dissecting the Structural Determinants of a Phenylalanine Aminomutase and Ammonia Lyase

January 20th, 2015 by Matthew M. Heberling, Marcelo F. Masman, Sebastian Bartsch, Gjalt G. Wybenga, Bauke W. Dijkstra, Siewert J. Marrink and Dick B. Janssen

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ACS Chemical Biology
DOI: 10.1021/cb500794h
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Selective Inhibitor of Platelet-Activating Factor Acetylhydrolases 1b2 and 1b3 That Impairs Cancer Cell Survival

January 20th, 2015 by Jae Won Chang, Andrea M. Zuhl, Anna E. Speers, Sherry Niessen, Steven J. Brown, Melinda M. Mulvihill, Yi Chiao Fan, Timothy P. Spicer, Mark Southern, Louis Scampavia, Virneliz Fernandez-Vega, Melissa M. Dix, Michael D. Cameron, Peter S. Hodder, Hugh

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ACS Chemical Biology
DOI: 10.1021/cb500893q
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Genetically Encoding Lysine Modifications on Histone H4

January 20th, 2015 by Bryan J. Wilkins, Liljan E. Hahn, Svenja Heitmüller, Holm Frauendorf, Oliver Valerius, Gerhard H. Braus and Heinz Neumann

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ACS Chemical Biology
DOI: 10.1021/cb501011v

Manganese and Microbial Pathogenesis: Sequestration by the Mammalian Immune System and Utilization by Microorganisms

January 16th, 2015 by Megan Brunjes Brophy and Elizabeth M. Nolan

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ACS Chemical Biology
DOI: 10.1021/cb500792b
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