A Small Molecule That Inhibits OGT Activity in Cells

March 18th, 2015 by Rodrigo F. Ortiz-Meoz, Jiaoyang Jiang, Michael B. Lazarus, Marina Orman, John Janetzko, Chenguang Fan, Damien Y. Duveau, Zhi-Wei Tan, Craig J. Thomas and Suzanne Walker

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00004

Constructing de Novo H2O2 Signaling via Induced Protein Proximity

March 18th, 2015 by Guihua Zeng, Roushu Zhang, Weimin Xuan, Wei Wang and Fu-Sen Liang

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00170

Optochemical Dissection of T-box Gene-Dependent Medial Floor Plate Development

March 17th, 2015 by Alexander Y. Payumo, Whitney J. Walker, Lindsey E. McQuade, Sayumi Yamazoe and James K. Chen

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ACS Chemical Biology
DOI: 10.1021/cb5010178

Identification and Validation of Novel Small Molecule Disruptors of HuR-mRNA Interaction

March 17th, 2015 by Xiaoqing Wu, Lan Lan, David Michael Wilson, Rebecca T. Marquez, Wei-chung Tsao, Philip Gao, Anuradha Roy, Benjamin Andrew Turner, Peter McDonald, Jon A Tunge, Steven A Rogers, Dan A. Dixon, Jeffrey AubeĢ and Liang Xu

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ACS Chemical Biology
DOI: 10.1021/cb500851u

Chemoenzymatically Prepared Heparan Sulfate Containing Rare 2-O-Sulfonated Glucuronic Acid Residues

March 17th, 2015 by Rio S. Boothello, Aurijit Sarkar, Vy My Tran, Thao Kim Nu Nguyen, Nehru Viji Sankaranarayanan, Akul Y. Mehta, AlHumaidi Alabbas, Spencer Brown, Alessandro Rossi, April C. Joice, Caitlin P. Mencio, Maritza V. Quintero, Balagurunathan Kuberan and Umesh

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00071
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Inhibitor Recognition Specificity of MERS-CoV Papain-like Protease May Differ from That of SARS-CoV

March 16th, 2015 by Hyun Lee, Hao Lei, Bernard D. Santarsiero, Joseph L. Gatuz, Shuyi Cao, Amy J. Rice, Kavankumar Patel, Michael Z. Szypulinski, Isabel Ojeda, Arun K. Ghosh and Michael E. Johnson

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ACS Chemical Biology
DOI: 10.1021/cb500917m
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Diazirine Photocrosslinking Recruits Activated FTO Demethylase Complexes for Specific N6-methyladenosine Recognition

March 16th, 2015 by Hyun Seok Jeong, Gosuke Hayashi and Akimitsu Okamoto

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ACS Chemical Biology
DOI: 10.1021/cb5010096
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Starter Unit Flexibility for Engineered Product Synthesis by the Nonreducing Polyketide Synthase PksA

March 10th, 2015 by Callie R. Huitt-Roehl, Eric A. Hill, Martina M. Adams, Anna L. Vagstad, Jesse W. Li and Craig A. Townsend

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00005
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Michael-Type Cyclizations in Lantibiotic Biosynthesis Are Reversible

March 10th, 2015 by Xiao Yang and Wilfred A. van der Donk

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00007

Chemically-Modified Peptides Targeting the PDZ Domain of GIPC as a Therapeutic Approach for Cancer

March 9th, 2015 by Chitta Ranjan Patra, Chamila N. Rupasinghe, Shamit K. Dutta, Santanu Bhattacharya, Enfeng Wang, Mark R. Spaller and Debabrata Mukhopadhyay

ACS Chemical Biology
DOI: 10.1021/cb500865a
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