A Note of Caution on the Role of Halogen Bonds for Protein Kinase/Inhibitor Recognition Suggested by High- And Low-Salt CK2α Complex Structures

May 15th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00235
  • Posted in ACS Chemical Biology, Publications
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Mad2 Inhibitor-1 (M2I-1): A Small Molecule Protein–Protein Interaction Inhibitor Targeting the Mitotic Spindle Assembly Checkpoint

May 15th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00121
  • Posted in ACS Chemical Biology, Publications
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A Genetically Encoded FRET Probe to Detect Intranucleosomal Histone H3K9 or H3K14 Acetylation Using BRD4, a BET Family Member

May 15th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/cb501046t
  • Posted in ACS Chemical Biology, Publications
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Incorporation of Unnatural Amino Acids in Response to the AGG Codon

May 12th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00230

Activity-Based Protein Profiling of Oncogene-Driven Changes in Metabolism Reveals Broad Dysregulation of PAFAH1B2 and 1B3 in Cancer

May 7th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00053
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Light-Activated Proteolysis for the Spatiotemporal Control of Proteins

May 7th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00069

Residue-Based Preorganization of BH3-Derived α/β-Peptides: Modulating Affinity, Selectivity and Proteolytic Susceptibility in α-Helix Mimics

May 7th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00109
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Anti-Group B Streptococcus Glycan-Conjugate Vaccines Using Pilus Protein GBS80 As Carrier and Antigen: Comparing Lysine and Tyrosine-directed Conjugation

May 6th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00247
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The Effect of Halogen-to-Hydrogen Bond Substitution on Human Aldose Reductase Inhibition

May 6th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00151

Formation of a Novel Macrocyclic Alkaloid from the Unnatural Farnesyl Diphosphate Analogue Anilinogeranyl Diphosphate by 5-Epi-Aristolochene Synthase

May 4th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00145
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