Optimized Plk1 PBD Inhibitors Based on Poloxin Induce Mitotic Arrest and Apoptosis in Tumor Cells

August 27th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00565
  • Posted in ACS Chemical Biology, Publications
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Binding Isotope Effects for para-Aminobenzoic Acid with Dihydropteroate Synthase from Staphylococcus aureus and Plasmodium falciparum

August 27th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00490
  • Posted in ACS Chemical Biology, Publications
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Direct Monitoring of Nucleotide Turnover in Human Cell Extracts and Cells by Fluorogenic ATP Analogs

August 23rd, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00459
  • Posted in ACS Chemical Biology, Publications
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Regulation of Proteasomal Degradation by Modulating Proteasomal Initiation Regions

August 21st, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00554

Position of Proline Mediates the Reactivity of S-Palmitoylation

August 19th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00429

Beyond a Fluorescent Probe: Inhibition of Cell Division Protein FtsZ by mant-GTP Elucidated by NMR and Biochemical Approaches

August 17th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00444
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A Small Molecule Inhibits Deregulated NRF2 Transcriptional Activity in Cancer

August 17th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00448

Leveraging the Mechanism of Oxidative Decay for Adenylate Kinase to Design Structural and Functional Resistances

August 17th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00431
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Virtual Screening for UDP-Galactopyranose Mutase Ligands Identifies a New Class of Antimycobacterial Agents

August 17th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00370
  • Posted in ACS Chemical Biology, Publications
  • Comments Off on Virtual Screening for UDP-Galactopyranose Mutase Ligands Identifies a New Class of Antimycobacterial Agents

Modifying an Insect Cell N-Glycan Processing Pathway Using CRISPR-Cas Technology

August 13th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00340