Evaluation of Kinase Activity Profiling Using Chemical Proteomics

October 5th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00616

Chemoproteomics Reveals Novel Protein and Lipid Kinase Targets of Clinical CDK4/6 Inhibitors in Lung Cancer

October 5th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00368
  • Posted in ACS Chemical Biology, Publications
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Experimental and Theoretical Evaluation of the Ethynyl Moiety as a Halogen Bioisostere

October 1st, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00515

Selective Targeting of Extracellular Insulin-Degrading Enzyme by Quasi-Irreversible Thiol-Modifying Inhibitors

September 30th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00334
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Mannoside Glycolipid Conjugates Display Anti-inflammatory Activity by Inhibition of Toll-like Receptor-4 Mediated Cell Activation

September 30th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00552
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MAP4K4 Is a Threonine Kinase That Phosphorylates FARP1

September 29th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00679

Studying a Drug-like, RNA-Focused Small Molecule Library Identifies Compounds That Inhibit RNA Toxicity in Myotonic Dystrophy

September 28th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00430
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Characterization of DDR2 Inhibitors for the Treatment of DDR2 Mutated Nonsmall Cell Lung Cancer

September 24th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00655

Antisense RNA-based High-Throughput Screen System for Directed Evolution of Quorum Quenching Enzymes

September 24th, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00714
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Chemical Proteomic Platform To Identify Citrullinated Proteins

September 23rd, 2015 by

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ACS Chemical Biology
DOI: 10.1021/acschembio.5b00438