Publisher Correction: BAF complex vulnerabilities in cancer demonstrated via structure-based PROTAC design
July 2nd, 2019 by William Farnaby
Nature Chemical Biology, Published online: 02 July 2019; doi:10.1038/s41589-019-0329-z
Publisher Correction: BAF complex vulnerabilities in cancer demonstrated via structure-based PROTAC designBAF complex vulnerabilities in cancer demonstrated via structure-based PROTAC design
June 10th, 2019 by William Farnaby
Nature Chemical Biology, Published online: 10 June 2019; doi:10.1038/s41589-019-0294-6
A structure-based design allows the development of a potent PROTAC to degrade BAF ATPase subunits SMARCA2 and SMARCA4 via recruitment of E3 ubiquitin ligase VHL and induce cancer cell death.