Structure-Guided DOT1L Probe Optimization by Label-Free Ligand Displacement
January 15th, 2015 by Joanna S. Yi, Alexander J. Federation, Jun Qi, Sirano Dhe-Paganon, Michael Hadler, Xiang Xu, Roodolph St. Pierre, Anthony C. Varca, Lei Wu, Jason J. Marineau, William B. Smith, Amanda Souza, Emma J. Chory, Scott A. Armstrong and James E. Bradner
ACS Chemical Biology
DOI: 10.1021/cb500796d